数字农科院2.0

Synthesis and Fungicidal Activities of Azaindolyl Thiazoline Compounds

文献类型： 外文期刊

作者： Xiao Yumei;Yuan Dekai;Zhang Zhenhua;Fu Bin;Yan Xiaojing;Yuan Huizhu

作者机构：

关键词： azaindolyl;thiazoline;synthesis;fungicidal activity

期刊名称： CHINESE JOURNAL OF ORGANIC CHEMISTRY

ISSN： 0253-2786

年卷期： 2016 年 36 卷 1 期

页码：

收录情况： SCI

摘要： In order to find new agrochemical products with high activities, 20 azaindolyl thiazoline compounds were designed and synthesized, and their structures were identified by spectral methods. At the concentration of 50 mg/L, some of the title compounds showed good fungicidal activities. Among those compounds, the EC50 values of 2a and 2d against Phomopsis asparagi and Pyricularia oryzae Cav are 6.55 and 9.66 mg/L, which are superior or comparable to the control pesticides, then they can serve as the lead compounds for new fungicide discovery.

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